Compound · citrus-bergamot
T2Supplement

Citrus Bergamot Extract

Polyphenol-rich extract from Citrus bergamia containing bergamottin, brutieridin, and melitidin. Brutieridin and melitidin are structural analogs of HMG-CoA reductase substrates, providing statin-like inhibition of cholesterol synthesis. Additionally activates AMPK in hepatocytes and inhibits pancreatic cholesterol ester transferase (ACAT), reducing intestinal cholesterol absorption.

Half-life
~6 hours (estimated from polyphenol PK)
Bioavailability
~30% (oral, polyphenol fraction)
Route
oral
Evidence tier
T2 — Single-RCT or mechanistic
Optimization pillars
cellular-health
References
2 peer-reviewed
Dose ranges

Three tiers ordered by aggressiveness. Tier chips on every OPTIMIZE intervention let you filter the catalog by your evidence tolerance.

conservative
500 mg/day
General cardiovascular support
moderate
500–1000 mg/day
Standard lipid management dose
aggressive
1000–1500 mg/day
Maximum studied dose for dyslipidemia
Monitoring
  • lipid-panel
  • hdl
  • ldl
  • triglycerides
  • apob
  • alt
  • ast
Contraindications
  • statin-interaction-monitor
References
  • PMID:23735317Bergamot polyphenolic fraction supplementation reduces lipid transfer protein levels in hyperlipidemic subjectsInt J Cardiol, 2013
  • PMID:26447646Hypolipidemic and antioxidant effects of bergamot polyphenol extract in patients with moderate hypercholesterolemiaFitoterapia, 2016
Notes

Citrus bergamot is the lipid management supplement for people who want statin-like effects without statins. The brutieridin and melitidin molecules structurally mimic HMG-CoA substrates — same mechanism as statins, weaker magnitude, but additive with other interventions. Clinical data shows 20-30% LDL reduction and 20-40% triglyceride reduction at 1000mg daily. Pairs well with berberine for a non-pharmaceutical lipid stack.

This is not medical advice

Discuss with a licensed clinician before starting, stopping, or changing any compound. This page documents what the research literature describes — it is not a prescription.

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