Compound · dutasteride
T1Pharmaceutical

Dutasteride

Dual inhibitor of both type I and type II 5-alpha reductase isoenzymes, reducing serum DHT by over 90%. The 5-week terminal half-life reflects extensive tissue binding and enterohepatic recirculation. More complete DHT suppression than finasteride but with correspondingly greater neurosteroid disruption.

Half-life
5 weeks
Bioavailability
60% (oral, increased with food)
Route
oral
Evidence tier
T1 — Multiple RCTs
Optimization pillars
recovery
References
2 peer-reviewed
Dose ranges

Three tiers ordered by aggressiveness. Tier chips on every OPTIMIZE intervention let you filter the catalog by your evidence tolerance.

conservative
0.5 mg/day
Standard BPH and hair loss dosing
moderate
0.5 mg EOD
Reduced frequency approach
aggressive
0.5 mg/day
Maximum dosing. Single dose formulation
Monitoring
  • total-testosterone
  • free-testosterone
  • dhea-s
  • estradiol
  • psa
  • alt
  • ast
Contraindications
  • pregnancy-exposure
  • hepatic-impairment
  • pediatric-use
References
  • PMID:17032385Dutasteride, a dual 5alpha-reductase inhibitor, for the treatment of benign prostatic hyperplasiaExpert Opin Pharmacother, 2006
  • PMID:16728986The importance of dual 5alpha-reductase inhibition in the treatment of male pattern hair lossJ Am Acad Dermatol, 2006
Notes

Dutasteride is the nuclear option in the 5-alpha reductase category. 90%+ DHT suppression versus finasteride 70%. Dual isoenzyme inhibition versus single. And a 5-week half-life that means once you take it, you are committed for months. There is no rapid washout. This molecule was designed for prostate volume reduction where maximum DHT suppression is the explicit goal. Using it for hair loss is a risk-benefit calculation that most practitioners get wrong by focusing exclusively on efficacy without weighting the neurosteroid consequences of near-total DHT elimination.

This is not medical advice

Discuss with a licensed clinician before starting, stopping, or changing any compound. This page documents what the research literature describes — it is not a prescription.

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