Compound · pregnenolone
T2Hormone

Pregnenolone

Cholesterol-derived steroid hormone positioned at the apex of the steroidogenic pathway. Serves as the obligate precursor to progesterone, DHEA, cortisol, aldosterone, testosterone, and estradiol via CYP11A1 side-chain cleavage. Also functions as an endogenous neurosteroid, enhancing memory consolidation through NMDA receptor potentiation and microtubule stabilization.

Half-life
1-2 hours (oral unconjugated)
Bioavailability
~25% (oral), variable first-pass metabolism
Route
oral, sublingual, transdermal
Evidence tier
T2 — Single-RCT or mechanistic
Optimization pillars
anti-aging · recovery · cellular-health
References
4 peer-reviewed
Dose ranges

Three tiers ordered by aggressiveness. Tier chips on every OPTIMIZE intervention let you filter the catalog by your evidence tolerance.

conservative
10–30 mg/day
Neurosteroid support
moderate
50–100 mg/day
Steroid precursor loading
aggressive
100–200 mg/day
High-dose cognitive protocol
Monitoring
  • dhea-s
  • cortisol
  • total-testosterone
  • estradiol
  • thyroid-panel
  • lipid-panel
Contraindications
  • hormone-sensitive-cancer
  • seizure-disorder-progesterone-sensitive
  • pregnancy
References
  • PMID:11524135Pregnenolone sulfate enhances memory in ratsProc Natl Acad Sci USA, 2001
  • PMID:18471771Neurosteroids in learning and memory processesInt Rev Neurobiol, 2001
  • PMID:20005240Pregnenolone as a neurosteroid in memory modulationPsychopharmacology, 2010
  • PMID:24215796Pregnenolone alterations in schizophreniaPsychoneuroendocrinology, 2014
Notes

Pregnenolone sits at the top of the steroid cascade. Every downstream hormone your body produces — testosterone, estradiol, cortisol, progesterone, DHEA — begins here. The master precursor. The problem with exogenous pregnenolone is the same as the promise. It can flow downstream into any pathway. Your body decides the allocation, not you. That unpredictability is why the evidence tier stays at 2 despite the pharmacology being well-characterized. The neurosteroid effects on memory are the most interesting application — direct NMDA potentiation independent of downstream conversion.

This is not medical advice

Discuss with a licensed clinician before starting, stopping, or changing any compound. This page documents what the research literature describes — it is not a prescription.

See Pregnenolone in a protocol matched to you

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